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New search Medicine profile Paracetamol

Clinical medicine profile

Paracetamol

Analgesic / Antipyretic (non-opioid)

OTC
Evidence state Source not available Reviewed 14 Aug 2026
Route
Oral, Rectal, Intravenous
Schedule
OTC
ATC
Not assigned
PPB status
registered
Patient advice Check interactions
Verification required

This profile needs source confirmation

A traceable source link is not attached to this profile. Confirm prescribing decisions against the current SmPC and Kenya STG/EML.

01 Risk first

Safety essentials

The information most likely to change a prescribing or dispensing decision.

Contraindications

  • Severe active hepatic disease / acute liver failure.
  • Hypersensitivity.
  • Chronic heavy alcohol use — use reduced maximum daily dose or avoid.

Precautions

  • Risk of severe hepatotoxicity in overdose.
  • Chronic high-dose use, malnutrition, enzyme-inducing drugs, and alcohol increase risk.
  • Check total daily intake from all sources.
02 Point of care

Dosing matrix

Population and organ-function guidance, shown together for faster comparison.

Adult

Orally or as supp: 0.5-1g after 4-6 hours to a max. 4g. Child:<3 months; 10mg/kg 3 months-1 year; 60-120mg, 6-12 years: 250-500mg. Repeated after 4-6 hours to max. of 4 doses in 24 hours. Parenteral: 10mg/kg body weight/dose given IV or deep IM after 4-6 hours to a max. of 5 doses (preferably not for more than 5 consecutive days).

Paediatric

Oral: 10–15 mg/kg/dose every 4–6 hours as needed. Maximum usually 60 mg/kg/day (do not exceed adult max). Use age/weight-appropriate formulations.

Renal

Severe renal impairment (e.g. CrCl <10–30 mL/min): increase dosing interval (e.g. every 6–8 hours) and avoid prolonged high doses; follow local protocol.

  • CrCl 30–120: Usual dosing if liver function normal; max 4 g/day adults.
  • CrCl 0–29: Consider 500–1000 mg every 6–8 h; avoid prolonged high doses; local protocol.
Hepatic

Avoid or use reduced dose in active liver disease / chronic alcohol use. Absolute caution in severe hepatic impairment — risk of acute liver failure in overdose.

03 Clinical use

Use, effects & interactions

Indications

  • Mild to moderate pain (headache, dental pain, musculoskeletal pain, dysmenorrhoea)
  • Clinical selection for Paracetamol should follow culture results where relevant, Kenya STG/EML recommendations, and the current product SmPC.
  • Class context: Analgesic / Antipyretic (non-opioid).
  • Confirm site-specific dose, duration and monitoring before prescribing.

Adverse effects

  • Rare at therapeutic doses.
  • Serious: acute liver failure in overdose, rare severe skin reactions (SJS/TEN/AGEP).
  • First-line for mild–moderate pain and fever.
  • Calculate total daily exposure from all sources.
  • In overdose: timed levels + NAC per protocol — do not wait for symptoms.
04 Pharmacology

Mechanism & disposition

Inhibitors of cyclo-oxygenase [COX-1 and COX-2] enzyme that catalyzes the conversion of arachidonic acid to PGH2.

Inhibit COX↓ ProstaglandinsAnalgesia / anti-inflammatory
Read complete mechanism

Inhibitors of cyclo-oxygenase [COX-1 and COX-2] enzyme that catalyzes the conversion of arachidonic acid to PGH2. Paracetamol inhibits central prostaglandin synthesis via effects on cyclo-oxygenase pathways (including COX-2 preferential central effects) and may engage serotonergic descending pathways. Antipyretic effect via hypothalamic heat-regulating centre. Minimal peripheral anti-inflammatory action.

Onset

Oral: ~30–60 minutes

Duration

4–6 hours

Route

Oral, Rectal, Intravenous

Metabolism

(glucuronidation/sulfation; minor CYP2E1 to NAPQI).

Half-life

~2–3 h (prolonged in overdose/liver disease).

05 Special populations

Pregnancy, lactation & diet

Pregnancy

Analgesic/antipyretic of choice in pregnancy when needed; use lowest effective dose/shortest duration.

Lactation

Compatible with breastfeeding at standard doses.

06 Kenya market

Brands & loaded prices

FromKES 20
MedianKES 230
Listings49
BrandManufacturerPackObserved price
Acimol suspension Universal Corporation Ltd Oral Suspension Unavailable
ADOL SUPP. Not recorded 125MG * 10 KES 318.02Daima Chemist price-list reference ↗ Source date not recorded · verify current price
ANAMOL Not recorded 120/5ML SUSP 100ML KES 150.50Daima Chemist price-list reference ↗ Source date not recorded · verify current price
ANAMOL MR TABS 10*S Not recorded — KES 322.50Daima Chemist price-list reference ↗ Source date not recorded · verify current price
AXAPARA INJECTION AXA PARENTERALS LTD Injection Unavailable
BRAVEMOL INTRAVENOUS INFUSION PHARMA SPECIALITIES LIMITED Solution For Infusion Unavailable
CALPOL INFANT SUSPENSION Not recorded 100ML KES 217.17Daima Chemist price-list reference ↗ Source date not recorded · verify current price
CETAMOL * DAIMA BIASHARA / Wholesale Import 60ML C/P NEW PICE KES 47.02Daima Chemist price-list reference ↗ Source date not recorded · verify current price
CIPLADON DAIMA BIASHARA / Wholesale Import 1000MG TABS 8*S KES 314.21daima_biashara_price_list
CURAMOL DAIMA BIASHARA / Wholesale Import 60ML KES 27.95Daima Chemist price-list reference ↗ Source date not recorded · verify current price
CURAMOL FIZZ 500 TABLETS DAWA LIMITED Effervescent Tablet Unavailable
CURAMOL FIZZ 1000 TABLETS DAWA LIMITED Effervescent Tablet Unavailable
CURAMOL SY Not recorded 100ML. KES 39.77Daima Chemist price-list reference ↗ Source date not recorded · verify current price
DENTAMOL TABS * 20`S Not recorded — KES 58.05Daima Chemist price-list reference ↗ Source date not recorded · verify current price
Efferalgan 500mg UPSA SAS Effervescent Tablet 500mg Unavailable
Efferalgan 1000mg UPSA SAS Effervescent Tablet 1000mg Unavailable
EFFERALGAN PAEDIATRIC 3%, oral solution UPSA SAS Syrup Unavailable
FEVADOL Not recorded 1G EFF TABS 8*S KES 319.81Daima Chemist price-list reference ↗ Source date not recorded · verify current price
FEVASTIN ET 500 TIL HEALTHCARE PVT LTD Effervescent Tablet Unavailable
FEVASTIN ET 1000 TIL HEALTHCARE PVT LTD Effervescent Tablet Unavailable
GESIC IV INFUSION NEXTGEN PHARMACEUTICALS (K) LTD Infusion Unavailable
KAREMOL TABLETS KAREMAX INDUSTRIAL LTD Tablet Unavailable
MICROMOL IV GOODMED PHARMARCY LTD Infusion Unavailable
Panadol P.O. Box 26773 - 00100 Nairobi Oral Drops, Powder For Suspension 20 Unavailable
PANADOL ADVANCE HALEON KENYA LIMITED Tablet Unavailable
PANADOL ADVANCE TABS 100*S Not recorded — KES 578.32Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PANADOL BABY & INFANT DAIMA BIASHARA / Wholesale Import 60ML KES 229.68Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PANADOL ELIXIR HALEON KENYA LIMITED Oral Suspension Unavailable
PANADOL EXTRA SOLUBLE 24*S Not recorded — KES 512.00Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PANADOL EXTRA TABS * 100 Not recorded — KES 722.89Daima Chemist price-list reference ↗ Source date not recorded · verify current price
Para-Denk 125 Suppos Denk Pharma Suppository Unavailable
PARAFAST DAIMA BIASHARA / Wholesale Import 1GM TABS 8*S KES 257.81Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PARAFAST ET DAIMA BIASHARA / Wholesale Import 500MG TABS 16*S KES 279.69Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PARAFAST ET JUNIOR Not recorded 160MG EFF TABS 10'S KES 247.25Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PARAFAST ET JUNIOR HighChem Marketing Ltd. Effervescent Tablet Unavailable
PARAGEN INJECTION P.O BOX 22953-00100 NAIROBI. Solution For Injection PARACETAMOL 1000MG/100ML (1%W/V) Unavailable
Paralife UNISEL LIMITED Injection Unavailable
PAROL DAIMA BIASHARA / Wholesale Import SYRUP 100ML KES 337.50Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PAROL TABS 30*S Not recorded — KES 193.50Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PHARMADOL Not recorded 500MG TABS 100*S KES 96.75Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PHARMADOL FIZZ Not recorded 500MG TABS 16*S KES 175.22Daima Chemist price-list reference ↗ Source date not recorded · verify current price
PHARMADOL FIZZ 500 GALAXY PHARMACEUTICAL LTD Effervescent Tablet Unavailable
PHARMADOL FIZZ 1000 GALAXY PHARMACEUTICAL LTD Effervescent Tablet Unavailable
SAVOEFFER Not recorded 1000MG EFF TABS 12*S KES 322.50Daima Chemist price-list reference ↗ Source date not recorded · verify current price
Tasamol Solution for Infusion Tasa Pharma Ltd Solution For Infusion Unavailable
TOTOMOL DAIMA BIASHARA / Wholesale Import 100ML KES 40.85Daima Chemist price-list reference ↗ Source date not recorded · verify current price
TOTOMOL SUSPENSION Not recorded 60ML KES 26.88Daima Chemist price-list reference ↗ Source date not recorded · verify current price
TRUMOL Not recorded 120MG/5ML SUSP 100ML KES 20.43Daima Chemist price-list reference ↗ Source date not recorded · verify current price
XYKAA EXTEND 30*S Not recorded — KES 645.00Daima Chemist price-list reference ↗ Source date not recorded · verify current price
07 Provenance

Sources & review state

Primary sourceLocal active-ingredient clinical extract; WHO Model Formulary / standard SmPC consensus (batch 1 research); Professional class pharmacology (Non-opioid analgesic / antipyretic)
Last reviewed14 Aug 2026
EvidenceSource not available

Decision support only. Confirm patient-specific decisions against the current product SmPC, Kenya STG/EML, and professional judgement.